Publications 2024
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Novel trends in homogenous and superwettable functional surfaces with a focus on siloxane and silane chemistry. PhD dissertation
Paulssen, D.
2024, August 22. Karlsruher Institut für Technologie (KIT). doi:10.5445/IR/1000171093/v2 -
Nanoliter Droplet Microarrays Combined with Impedance Spectroscopy and Sandwiching Method for Advancements in Miniaturized Cell Culture and Screening. PhD dissertation
Zhou, M.
2024, August 19. Karlsruher Institut für Technologie (KIT). doi:10.5445/IR/1000172875 -
Design and Synthesis of New Dihydropyrimidine Derivatives with a Cytotoxic Effect as Dual EGFR/VEGFR-2 Inhibitors
Al-Wahaibi, L. H.; Elshamsy, A. M.; Ali, T. F. S.; Youssif, B. G. M.; Bräse, S.; Abdel-Aziz, M.; El-Koussi, N. A.
2024. ACS Omega, 9 (32), 34358–34369. doi:10.1021/acsomega.4c01361 -
New Diaryl-1,2,4-triazolo[3,4- a ]pyrimidine Hybrids as Selective COX-2/sEH Dual Inhibitors with Potent Analgesic/Anti-inflammatory and Cardioprotective Properties
Al-Wahaibi, L. H.; Abdel-Rahman, M. H.; El-Adl, K.; Youssif, B. G. M.; Bräse, S.; Abdel-Aziz, S. A.
2024. ACS Omega, 9 (31), 33494–33509. doi:10.1021/acsomega.4c00870 -
Key role of cycloalkyne nature in alkyne-dye reagents for enhanced specificity of intracellular imaging by bioorthogonal bioconjugation
Vidyakina, A. A.; Silonov, S. A.; Govdi, A. I.; Ivanov, A. Y.; Podolskaya, E. P.; Balova, I. A.; Bräse, S.; Danilkina, N. A.
2024. Organic & Biomolecular Chemistry. doi:10.1039/d4ob01032a -
Convenient synthesis and X-ray determination of 2-amino-6 H -1,3,4-thiadiazin-3-ium bromides endowed with antiproliferative activity
Tawfeek, H. N.; Abdelmoez, A.; Dahlous, K. A.; Youssif, B. G. M.; Bräse, S.; Rissanen, K.; Nieger, M.; El-Sheref, E. M.
2024. RSC Advances, 14 (25), 17866 – 17876. doi:10.1039/D4RA02531H -
3D printing of reactive macroporous polymers via thiol–ene chemistry and polymerization-induced phase separation
Mandsberg, N. K.; Aslan, F.; Dong, Z.; Levkin, P. A.
2024. Chemical Communications, 60 (45), 5872 – 5875. doi:10.1039/D4CC00466C -
Thio-2 Inhibits Key Signaling Pathways Required for the Development and Progression of Castration-resistant Prostate Cancer
Neeb, A.; Figueiredo, I.; Bogdan, D.; Cato, L.; Stober, J.; Jiménez-Vacas, J. M.; Gourain, V.; Lee, I. I.; Seeger, R.; Muhle-Goll, C.; Gurel, B.; Welti, J.; Nava Rodrigues, D.; Rekowski, J.; Qiu, X.; Jiang, Y.; Di Micco, P.; Mateos, B.; Bielskutė, S.; Riisnaes, R.; Ferreira, A.; Miranda, S.; Crespo, M.; Buroni, L.; Ning, J.; Carreira, S.; Bräse, S.; Jung, N.; Gräßle, S.; Swain, A.; Salvatella, X.; Plymate, S. R.; Al-Lazikani, B.; Long, H. W.; Yuan, W.; Brown, M.; Cato, A. C. B.; de Bono, J. S.; Sharp, A.
2024. Molecular Cancer Therapeutics, 23 (6), 791–808. doi:10.1158/1535-7163.MCT-23-0354 -
Discovery of new Schiff bases of the disalicylic acid scaffold as DNA gyrase and topoisomerase IV inhibitors endowed with antibacterial properties
Al-Wahaibi, L. H.; Mahmoud, M. A.; Alzahrani, H. A.; Abou-Zied, H. A.; Gomaa, H. A. M.; Youssif, B. G. M.; Bräse, S.; Rabea, S. M.
2024. Frontiers in Chemistry, 12, Art.-Nr.: 1419242. doi:10.3389/fchem.2024.1419242 -
A New Class of Chiral Polyethers and Polyesters Based on the [2.2]Paracyclophane Scaffold
Kern, P.; Tappert, H.; Bräse, S.
2024. Polymers, 16 (11), Art.-Nr.: 1603. doi:10.3390/polym16111603 -
Substituted Pyrrole‐based Schiff Bases: Effect On The Luminescence Of Neutral Heteroleptic Cu(I) Complexes
Ferraro, V.; Fuhr, O.; Bizzarri, C.; Bräse, S.
2024. European Journal of Inorganic Chemistry, 27 (17), Art.-Nr.: e202400080. doi:10.1002/ejic.202400080 -
Application of High-Throughput Screenings on the Interfaces of Chemistry, Biology and Material Science. PhD dissertation
Seifermann, M.
2024, May 14. Karlsruher Institut für Technologie (KIT). doi:10.5445/IR/1000168798 -
Parallel and Miniaturized Combinatorial Synthesis and Analysis of Small Molecules on Droplet Microarray. PhD dissertation
Höpfner, J.
2024, May 14. Karlsruher Institut für Technologie (KIT). doi:10.5445/IR/1000168797 -
Miniaturized Chemistry: from Synthesis in Nanoliters to Purification and High-Throughput Screening. PhD dissertation
Wiedmann, J. J.
2024, March 26. Karlsruher Institut für Technologie (KIT). doi:10.5445/IR/1000166093 -
Reversing the stereoselectivity of intramolecular [2+2] photocycloaddition utilizing cucurbit[8]uril as a molecular flask
Qiu, X.; Seibert, J.; Fuhr, O.; Biedermann, F.; Bräse, S.
2024. Chemical Communications, 60 (24), 3267–3270. doi:10.1039/D3CC05783F -
Stereoselective synthesis and X-ray structure determination of novel 1,2-dihydroquinolinehydrazonopropanoate derivatives
Tawfeek, H. N.; Tawfeek, A. M.; Bräse, S.; Nieger, M.; El-Sheref, E. M.
2024. Heliyon, 10 (4), Art.-Nr.: e25248. doi:10.1016/j.heliyon.2024.e25248 -
Optimized Detection of Volatile Organic Compounds Utilizing Durable and Selective Arrays of Tailored UiO-66-X SURMOF Sensors
Okur, S.; Hashem, T.; Bogdanova, E.; Hodapp, P.; Heinke, L.; Bräse, S.; Wöll, C.
2024. ACS Sensors, 9 (2), 622–630. doi:10.1021/acssensors.3c01575 -
ANDeS: An automated nanoliter droplet selection and collection device
Urrutia Gómez, J. E.; Faraj, R. E. K. E.; Braun, M.; Levkin, P. A.; Popova, A. A.
2024. SLAS Technology, 29 (1), Art.-Nr.: 100118. doi:10.1016/j.slast.2023.11.002 -
From Mono- to Polynuclear 2-(Diphenylphosphino)pyridine-Based Cu(I) and Ag(I) Complexes: Synthesis, Structural Characterization, and DFT Calculations
Busch, J. M.; Rehak, F. R.; Ferraro, V.; Nieger, M.; Kemell, M.; Fuhr, O.; Klopper, W.; Bräse, S.
2024. ACS Omega, 9 (2), 2220–2233. doi:10.1021/acsomega.3c05755 -
Synthesis of substituted triazole–pyrazole hybrids using triazenylpyrazole precursors
Gräßle, S.; Holzhauer, L.; Wippert, N.; Fuhr, O.; Nieger, M.; Jung, N.; Bräse, S.
2024. Beilstein Journal of Organic Chemistry, 20, 1396 – 1404. doi:10.3762/bjoc.20.121 -
CART: Carrier‐Based Actuatable and Reprogrammable Transport
Mandsberg, N. K.; Serna, J. A.; Levkin, P. A.
2024. Advanced Functional Materials, 2406635. doi:10.1002/adfm.202406635 -
High-throughput screening for cell binding and repulsion peptides on multifunctionalized surfaces
Sonnentag, S. J.; Jenne, F.; Orian-Rousseau, V.; Nesterov-Mueller, A.
2024. Communications Biology, 7 (1), Art.-Nr.: 870. doi:10.1038/s42003-024-06541-7 -
(Semi-) Automatic Review Process for Common Compound Characterization Data in Organic Synthesis
Huang, Y.-C.; Tremouilhac, P.; Kuhn, S.; Huang, P.-C.; Lin, C.-L.; Schlörer, N.; Taubert, O.; Götz, M.; Jung, N.; Bräse, S.
2024. ChemRxiv. doi:10.26434/chemrxiv-2024-1r9tb -
Thermally Activated Delayed Fluorescence (TADF) Materials Based on Earth‐Abundant Transition Metal Complexes: Synthesis, Design and Applications
Ferraro, V.; Bizzarri, C.; Bräse, S.
2024. Advanced Science, 2404866. doi:10.1002/advs.202404866 -
Effect of tert-butyl substitution on controlling the orientation of TADF emitters in guest–host systems
Sahay, P.; Crovini, E.; Stavrou, K.; Zhang, Z.; Nguyên, B. M.; Wagner, D.; Strohriegl, P.; Bräse, S.; Monkman, A.; Zysman-Colman, E.; Brütting, W.
2024. Journal of Materials Chemistry C. doi:10.1039/D4TC01195C -
Enhancing Temperature Responsiveness of PNIPAM Through 3D‐Printed Hierarchical Porosity
Liu, W.; Wang, Z.; Serna, J. A.; Debastiani, R.; Gomez, J. E. U.; Lu, L.; Yang, W.; Dong, Z.; Levkin, P. A.
2024. Advanced Functional Materials, Artkl.Nr.: 2403794. doi:10.1002/adfm.202403794 -
From Molecules to Materials: Collaborative Research at the Chemistry—Materials Science Interface and Lessons Learned in Cyclophane Chemistry
Hassan, Z.; Zysman-Colman, E.; Lahann, J.; Bräse, S.
2024. Advanced Functional Materials, Art.-Nr.: 202403365. doi:10.1002/adfm.202403365 -
Doping Strategies for Tetrasubstituted Paracyclophane Hole Transport Layers in Perovskite Solar Cells
Schulz, A. D.; Otterbach, S. A.; Tappert, H.; Elsing, D.; Wenzel, W.; Kozlowska, M.; Bräse, S.; Colsmann, A.; Röhm, H.
2024. Advanced Functional Materials, Art.-Nr.: 2402110. doi:10.1002/adfm.202402110 -
Modulation of neuroinflammation and oxidative stress by targeting GPR55 – new approaches in the treatment of psychiatric disorders
Apweiler, M.; Saliba, S. W.; Sun, L.; Streyczek, J.; Normann, C.; Hellwig, S.; Bräse, S.; Fiebich, B. L.
2024. Molecular Psychiatry. doi:10.1038/s41380-024-02614-5 -
Design and synthesis of new dihydropyrimidine/sulphonamide hybrids as promising anti-inflammatory agents via dual mPGES-1/5-LOX inhibition
Al-Wahaibi, L. H.; Elshamsy, A. M.; Ali, T. F. S.; Youssif, B. G. M.; Bräse, S.; Abdel-Aziz, M.; El-Koussi, N. A.
2024. Frontiers in Chemistry, 12, Art.-Nr.: 1387923. doi:10.3389/fchem.2024.1387923 -
Extraction of the intrinsic rate constant for a photocyclization reaction in capillary microreactors using a simplified reactor model
Li, J.; Šimek Tosino, H.; Ladewig, B. P.; Jung, N.; Bräse, S.; Dittmeyer, R.
2024. Reaction Chemistry & Engineering. doi:10.1039/d4re00087k -
Targeting CD44 and other pleiotropic co-receptors as a means for broad inhibition of tumor growth and metastasis
Mehner, L.-M.; Munoz-Sagredo, L.; Sonnentag, S. J.; Treffert, S. M.; Orian-Rousseau, V.
2024. Clinical and Experimental Metastasis. doi:10.1007/s10585-024-10292-4 -
Linker aggregation engineering of TADF materials to tune carrier balance for highly efficient organic LEDs with long operational lifetime
Zhang, Z.; Xia, R.; Wang, K.; Wu, Y.; Zang, P.; Gan, X.; Liao, Z.; Wei, B.; Wu, P.; Bräse, S.; Wang, Z.
2024. Aggregate, Art.-Nr.: e588. doi:10.1002/agt2.588 -
Solvent‐Independent 3D Printing of Organogels
Kuzina, M. A.; Hoffmann, M.; Mandsberg, N. K.; Domínguez, C. M.; Niemeyer, C. M.; Wilhelm, M.; Levkin, P. A.
2024. Advanced Functional Materials, Art.-Nr.: 2403694. doi:10.1002/adfm.202403694 -
Anti-Neuroinflammatory Effects of a Macrocyclic Peptide-Peptoid Hybrid in Lipopolysaccharide-Stimulated BV2 Microglial Cells
Sun, L.; Wilke Saliba, S.; Apweiler, M.; Akmermer, K.; Herlan, C.; Grathwol, C.; de Oliveira, A. C. P.; Normann, C.; Jung, N.; Bräse, S.; Fiebich, B. L.
2024. International Journal of Molecular Sciences, 25 (8), Artkl.Nr.:4462. doi:10.3390/ijms25084462 -
A Novel Carbazolophane: A Comparison of the Performance of Two Planar Chiral CP‐TADF Emitters
Seibert, J.; Xu, Y.; Hafeez, H.; Podlech, J.; Favereau, L.; Spuling, E.; Waldhelm, C.; Nieger, M.; Fuhr, O.; Hassan, Z.; Crassous, J.; Samuel, I. D. W.; Zysman-Colman, E.; Bräse, S.
2024. Advanced Functional Materials, Art.-Nr.: 2401956. doi:10.1002/adfm.202401956 -
Synthetic methodology of pyrimido[4,5‐ b ]quinoline derivatives
Tawfeek, H. N.; Hasanin, T. H. A.; Bräse, S.
2024. Journal of Heterocyclic Chemistry, 61 (6), 971–1008. doi:10.1002/jhet.4815 -
Modulating and Accelerating Photolysis of Photoactivatable [2.2]Paracyclophane Aryl Azide in Supramolecular Host for Bioimaging
Qiu, X.; Pohl, E.; Cai, Q.; Seibert, J.; Li, Y.; Leopold, S.; Fuhr, O.; Meier, M. A. R.; Schepers, U.; Bräse, S.
2024. Advanced Functional Materials, Art.-Nr.: 2401938. doi:10.1002/adfm.202401938 -
Synthesis of Mono‐, Di‐, Tri‐, and Tetra‐cationic Pyridinium and Vinylpyridinium Modified [2.2]Paracyclophanes: Modular Receptors for Supramolecular Systems
Wang, Y.; Li, Y.; Fuhr, O.; Nieger, M.; Hassan, Z.; Bräse, S.
2024. ChemistryOpen, 13 (8), e202400024. doi:10.1002/open.202400024 -
Wetting Behavior of Inkjet-Printed Electronic Inks on Patterned Substrates
Arya, P.; Wu, Y.; Wang, F.; Wang, Z.; Cadilha Marques, G.; Levkin, P. A.; Nestler, B.; Aghassi-Hagmann, J.
2024. Langmuir, 40 (10), 5162–5173. doi:10.1021/acs.langmuir.3c03297 -
Design, synthesis, and apoptotic antiproliferative action of new 1,2,3-triazole/1,2,4-oxadiazole hybrids as dual EGFR/VEGFR-2 inhibitors
Mahmoud, M. A.; Mohammed, A. F.; Salem, O. I. A.; Almutairi, T. M.; Bräse, S.; Youssif, B. G. M.
2024. Journal of Enzyme Inhibition and Medicinal Chemistry, 39 (1), Art.-Nr.: 2305856. doi:10.1080/14756366.2024.2305856 -
Constructing [2.2]Paracyclophane‐Based Ultrasensitive Optical Fluorescent‐Phosphorescent Thermometer with Cucurbit[8]uril Supramolecular Assembly
Qiu, X.; Zheng, T.; Runowski, M.; Woźny, P.; Martín, I. R.; Soler-Carracedo, K.; Piñero, C. E.; Lebedkin, S.; Fuhr, O.; Bräse, S.
2024. Advanced Functional Materials, Art.-Nr.: 2313517. doi:10.1002/adfm.202313517 -
Benzimidazole-Based Derivatives as Apoptotic Antiproliferative Agents: Design, Synthesis, Docking, and Mechanistic Studies
Youssif, B. G. M.; Morcoss, M. M.; Bräse, S.; Abdel-Aziz, M.; Abdel-Rahman, H. M.; Abou El-Ella, D. A.; Abdelhafez, E. S. M. N.
2024. Molecules, 29 (2), Art.-Nr.: 446. doi:10.3390/molecules29020446 -
High‐Throughput Miniaturized Synthesis of PROTAC‐Like Molecules
Tian, Y.; Seifermann, M.; Bauer, L.; Luchena, C.; Wiedmann, J. J.; Schmidt, S.; Geisel, A.; Afonin, S.; Höpfner, J.; Brehm, M.; Liu, X.; Hopf, C.; Popova, A. A.; Levkin, P. A.
2024. Small, Art.-Nr.: 2307215. doi:10.1002/smll.202307215 -
Azide Thermolysis Frameworks: Self‐inflating, Porous, and Lightweight Materials
Brückel, J.; Matt, Y.; Schmidt, L.; Mattern, C. M.; Schepers, U.; Leopold, S.; Calkovsky, M.; Gerthsen, D.; Bräse, S.
2024. ChemNanoMat, 10 (2), Art.-Nr.: e202300222. doi:10.1002/cnma.202300222 -
Modulating Aryl Azide Photolysis: Synthesis of a Room‐Temperature Phosphorescent Carboline in Cucurbit[7]uril Host
Qiu, X.; Wang, Y.; Leopold, S.; Lebedkin, S.; Schepers, U.; Kappes, M. M.; Biedermann, F.; Bräse, S.
2024. Small, 20 (16), Art.Nr.: 2307318. doi:10.1002/smll.202307318 -
Quantitative live imaging reveals a direct interaction between CD44v6 and MET in membrane domains upon activation with both MET ligands, HGF and internalin B
Tannoo, R. M.; Richert, L.; Koschut, D.; Tomishige, N.; Treffert, S. M.; Kobayashi, T.; Mély, Y.; Orian-Rousseau, V.
2024. Biochimica et Biophysica Acta (BBA) - Biomembranes, 1866 (1), Art.-Nr. 184236. doi:10.1016/j.bbamem.2023.184236 -
High‐Performance Pressure Sensors Based on Shaped Gel Droplet Arrays
Wang, Z.; Cai, Q.; Lu, L.; Levkin, P. A.
2024. Small, 20 (5), Art.Nr.: 2305214. doi:10.1002/smll.202305214 -
Palladium‐Catalyzed Combinatorial Synthesis of Biphenyls on Droplet Microarrays at Nanoliter Scale
Höpfner, J.; Brehm, M.; Levkin, P. A.
2024. Small, 20 (4), Art.Nr.: 2304325. doi:10.1002/smll.202304325 -
The Impact of Digitalized Data Management on Materials Systems Workflows
Tristram, F.; Jung, N.; Hodapp, P.; Schröder, R. R.; Wöll, C.; Bräse, S.
2024. Advanced Functional Materials, 34 (20), Art.-Nr.: 2303615. doi:10.1002/adfm.202303615 -
Disulfide‐Bridged Dynamic Covalent Triazine Polymer Thin Films by Interface Polymerization: High Refractive Index with Excellent Optical Transparency
Begum, S.; Kutonova, K.; Mauri, A.; Koenig, M.; Chan, K. C.; Sprau, C.; Dolle, C.; Trouillet, V.; Hassan, Z.; Leonhard, T.; Heißler, S.; Eggeler, Y. M.; Wenzel, W.; Kozlowska, M.; Bräse, S.
2024. Advanced Functional Materials, 34 (20), Art.-Nr.: 2303929. doi:10.1002/adfm.202303929 -
Functional Material Systems Enabled by Automated Data Extraction and Machine Learning
Kalhor, P.; Jung, N.; Bräse, S.; Wöll, C.; Tsotsalas, M.; Friederich, P.
2024. Advanced Functional Materials, 34 (20), Art.Nr.: 2302630. doi:10.1002/adfm.202302630 -
Recent Advances of Transition Metal Complexes for Photopolymerization and 3D Printing under Visible Light
Ferraro, V.; Adam, C. R.; Vranic, A.; Bräse, S.
2024. Advanced Functional Materials, 34 (20), Art.-Nr.: 2302157. doi:10.1002/adfm.202302157 -
Selective Peptide Binders to the Perfluorinated Sulfonic Acid Ionomer Nafion
Schmidt, D.; Gartner, P.; Berezkin, I.; Rudat, J.; Bilger, M.; Grünert, T.; Zimmerer, N.; Quarz, P.; Scharfer, P.; Brückel, J.; Jung, A. P.; Singh, P.; Pooja, P.; Meier, B.; Stahlberger, M.; Schabel, W.; Bräse, S.; Lanza, G.; Nesterov-Mueller, A.
2024. Advanced Functional Materials, 34 (20), Article no: 2214932. doi:10.1002/adfm.202214932 -
Exploring Functional Photonic Devices made from a Chiral Metal–Organic Framework Material by a Multiscale Computational Method
Zerulla, B.; Li, C.; Beutel, D.; Oßwald, S.; Holzer, C.; Bürck, J.; Bräse, S.; Wöll, C.; Fernandez-Corbaton, I.; Heinke, L.; Rockstuhl, C.; Krstić, M.
2024. Advanced Functional Materials, 34 (20), Art.-Nr.: 2301093. doi:10.1002/adfm.202301093 -
Tough PEGgels by In Situ Phase Separation for 4D Printing
Wang, Z.; Heck, M.; Yang, W.; Wilhelm, M.; Levkin, P. A.
2024. Advanced Functional Materials, 34 (20), Art.-Nr.: 2300947. doi:10.1002/adfm.202300947